Glycine receptor antagonist
A glycine receptor antagonist is a drug which acts as an antagonist of the glycine receptor.[1][2]
Examples
Antagonists
- Selective
- Brucine
- Strychnine
- Tutin
- Non-selective
- Bicuculline
- Caffeine
- Picrotoxin
- Pitrazepin
- Thiocolchicoside
See also
- Glycine receptor agonist
References
- ^ Miyakawa, N; Uchino, S; Yamashita, T; Okada, H; Nakamura, T; Kaminogawa, S; Miyamoto, Y; Hisatsune, T (16 September 2002). "A glycine receptor antagonist, strychnine, blocked NMDA receptor activation in the neonatal mouse neocortex". NeuroReport. 13 (13): 1667–73. doi:10.1097/00001756-200209160-00020. PMID 12352624. S2CID 34027498.
- ^ Vandenberg, RJ; Handford, CA; Schofield, PR (September 1992). "Distinct agonist- and antagonist-binding sites on the glycine receptor". Neuron. 9 (3): 491–6. doi:10.1016/0896-6273(92)90186-h. PMID 1326295. S2CID 45100334.
External links
- Media related to Glycine receptor antagonists at Wikimedia Commons
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Pharmacomodulation
- ♦ Enzyme: Inducer
- Inhibitor
- ♦ Ion channel: Opener
- Blocker
- ♦ Receptor: Agonist
- Partial agonist
- Antagonist
- Inverse agonist
- Positive allosteric modulator (PAM)
- Negative allosteric modulator (NAM)
- ♦ Miscellaneous: Precursor
- Cofactor
Enzyme | see Enzyme inhibition |
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Ion channel | See Ion channel modulators |
Receptor & transporter | |
Miscellaneous |
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